PROTAC BRD4 ligand-1
PROTAC BRD4 ligand-1 serves as the BRD4-targeting component of the PROTAC molecule GNE-987 and functions as a BET bromodomain inhibitor. This compound is utilized in chemical biology and oncology research to study targeted protein degradation, with applications in both cellular and in vivo models of cancer and inflammatory diseases.
Product Specifications
CAS Number
2313230-51-0
Product Name Alternative
BET, BRD4, LigandsforTargetProteinforPROTAC, Ligands for Target Protein for PROTAC, Epigenetic Reader Domain, EpigeneticReaderDomain, PROTAC BRD4 ligand 1, PROTAC BRD4 ligand1, PROTAC BRD4 ligand-1, PROTAC BRD-4 ligand-1
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Purity
99.28% (May vary between batches)
Solubility
DMSO:4.5 mg/mL (8.99 mM)
Smiles
Cn1cc2-c3cc (CS (C) (=O) =O) c (cc3N (Cc3c[nH]c (c23) c1=O) c1ncc (F) cc1F) C (O) =O
Molecular Formula
C23H18F2N4O5S
Molecular Weight
500.47
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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