Sitaxsentan
Sitaxsentan (TBC-11251) is a selective endothelin A (ETA) receptor antagonist that inhibits the potent vasoconstrictor endothelin. It is used in research for pulmonary arterial hypertension, with applications in both in vitro binding assays and in vivo hemodynamic studies.
Product Specifications
CAS Number
184036-34-8
Product Name Alternative
IPI1040, IPI-1040, IPI 1040, Endothelin Receptor, Endothelin A receptor, EndothelinReceptor, Sitaxsentan, TBC 11251, TBC11251, TBC-11251
Field of Research
Pharmacology & Drug Discovery
Purity
97.99% (May vary between batches)
Solubility
DMSO:4.55 mg/mL (10 mM)
Smiles
C (CC=1C=C2C (=CC1C) OCO2) (=O) C3=C (S (NC4=C (Cl) C (C) =NO4) (=O) =O) C=CS3
Molecular Formula
C18H15ClN2O6S2
Molecular Weight
454.9
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog