SSTR5 antagonist 1

SSTR5 antagonist 1 is a potent, orally bioavailable small molecule that selectively inhibits somatostatin receptor subtype 5. It demonstrates high affinity for human and mouse SSTR5 (IC50 = 9.6 and 57 nM, respectively) . This antagonist is a valuable research tool for investigating SSTR5 function in metabolic and endocrine studies, both in vitro and in vivo.