ZEN-3862
ZEN-3862 (Willardiine) is a potent, dual-bromodomain BET inhibitor with IC50 values of 0.16 μM and 0.13 μM for BRD4 (BD1) and BRD4 (BD2), respectively. This small molecule serves as a versatile ligand for constructing PROTAC degraders to selectively deplete BRD4 protein levels in cellular and biochemical research.
Product Specifications
CAS Number
1952264-33-3
Product Name Alternative
EpigeneticReaderDomain, Epigenetic Reader Domain, BRD4BD1, BRD4-BD2, BRD4 BD2, BD1-BRD4, ZEN 3862, ZEN3862, ZEN-3862
Field of Research
Epigenetics & Chromatin
Purity
97.10% (May vary between batches)
Solubility
DMSO:Soluble
Smiles
CC=1C (C2=CN (CC3=CC (F) =C (C=C3) C4CO4) C (=O) C=C2) =C (C) ON1
Molecular Formula
C19H17FN2O3
Molecular Weight
340.35
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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