ZEN-3862
ZEN-3862 (Willardiine) is a potent, dual-bromodomain BET inhibitor with IC50 values of 0.16 μM and 0.13 μM for BRD4 (BD1) and BRD4 (BD2), respectively. This small molecule serves as a versatile ligand for constructing PROTAC degraders to selectively deplete BRD4 protein levels in cellular and biochemical research.
Product Specifications
CAS Number
1952264-33-3
Product Name Alternative
EpigeneticReaderDomain, Epigenetic Reader Domain, BRD4BD1, BRD4-BD2, BRD4 BD2, BD1-BRD4, ZEN 3862, ZEN3862, ZEN-3862
Field of Research
Epigenetics & Chromatin
Purity
97.10% (May vary between batches)
Solubility
DMSO:Soluble
Smiles
CC=1C (C2=CN (CC3=CC (F) =C (C=C3) C4CO4) C (=O) C=C2) =C (C) ON1
Molecular Formula
C19H17FN2O3
Molecular Weight
340.35
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1449524-01 0.05 mg (E-Coli)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details MBS1449524-02 0.05 mg (Yeast)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details MBS1449524-03 0.2 mg (E-Coli)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details MBS1449524-04 0.5 mg (E-Coli)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details MBS1449524-05 0.05 mg (Baculovirus)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details MBS1449524-06 0.2 mg (Yeast)
Recombinant Buchnera aphidicola subsp. Acyrthosiphon pisum Anthranilate synthase component 2 (trpG)
Sign In for Pricing
View Details