CCG258208
GRKs-IN-1 is a potent and selective small molecule inhibitor, demonstrating high activity against GRK2 (IC50 = 130 nM) and moderate activity against GRK5 (IC50 = 7.1 μM) . This compound is a valuable research tool for investigating GRK2/5 signaling pathways in cardiovascular and oncology research, applicable in both cellular and biochemical assays.
Product Specifications
CAS Number
2055990-90-2
Field of Research
Pharmacology & Drug Discovery
Smiles
C (OC=1C=C2C (=CC1) OCO2) [C@H]3[C@@H] (CCNC3) C4=CC (C (NCC=5C=CNN5) =O) =C (F) C=C4
Molecular Formula
C24H25FN4O4
Molecular Weight
452.48
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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