CCG258208
GRKs-IN-1 is a potent and selective small molecule inhibitor, demonstrating high activity against GRK2 (IC50 = 130 nM) and moderate activity against GRK5 (IC50 = 7.1 μM) . This compound is a valuable research tool for investigating GRK2/5 signaling pathways in cardiovascular and oncology research, applicable in both cellular and biochemical assays.
Product Specifications
CAS Number
2055990-90-2
Field of Research
Pharmacology & Drug Discovery
Smiles
C (OC=1C=C2C (=CC1) OCO2) [C@H]3[C@@H] (CCNC3) C4=CC (C (NCC=5C=CNN5) =O) =C (F) C=C4
Molecular Formula
C24H25FN4O4
Molecular Weight
452.48
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
bs-18128R-BF488 100 µL
Phospho-IKB alpha (Ser32) Polyclonal Antibody, AbBy Fluor™ 488 Conjugated
Sign In for Pricing
View Details MK1F83-01 48 Test
Bovine Adenovirus 3 (BAdV-3) Probe-based qPCR Kit
Sign In for Pricing
View Details MK1F83-02 50 Tests
Bovine Adenovirus 3 (BAdV-3) Probe-based qPCR Kit
Sign In for Pricing
View Details ![ELK1 Antibody [7E10D5 / 7E10E8]](https://cdn.genprice.uk/genprice/uk/genprice4.webp)
14082-05021 150 µg
Canine Myoglobin (Mb) Antibody (Biotin Conjugate)
Sign In for Pricing
View Details