GSK8814
GSK8814 is a potent and selective chemical probe targeting the ATAD2/ATAD2B bromodomains, with a pKd of 8.1 and over 500-fold selectivity versus BRD4 BD1. This inhibitor is a valuable tool for investigating the role of ATAD2 in oncology research, supporting both in vitro mechanistic studies and in vivo model validation.
Product Specifications
CAS Number
1997369-78-4
Field of Research
Epigenetics & Chromatin
Smiles
CO[C@H]1CNC[C@@H] (OCC2CCC (F) (F) CC2) [C@@H]1Nc1ncc (-c2cncc (C) c2) c2cc (C) c (=O) [nH]c12
Molecular Formula
C28H35F2N5O3
Molecular Weight
527.61
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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