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K134

K134 is a selective phosphodiesterase 3 (PDE3) inhibitor, exhibiting potent activity against PDE3A and PDE3B with IC50 values of 0.1 and 0.28 μM, respectively, while showing significantly lower potency against PDE5, PDE2, and PDE4. This small molecule is a valuable research tool for investigating cAMP-mediated signaling pathways in cardiovascular, metabolic, and platelet function studies, applicable in both in vitro and in vivo experimental models.

Product Specifications

CAS Number

189362-06-9

Field of Research

Metabolism Research

Smiles

O[C@@H]1CCCC[C@H]1N (C1CC1) C (=O) NCCCOc1ccc2[nH]c (=O) ccc2c1

Molecular Formula

C22H29N3O4

Molecular Weight

399.48

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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