PF-02575799
PF-02575799 is a potent and selective small molecule inhibitor of microsomal triglyceride transfer protein (MTP), exhibiting an IC50 of 0.77±0.29 nM. This compound is a valuable research tool for investigating lipid metabolism, enabling in vitro and in vivo studies related to dyslipidemia and atherosclerosis.
Product Specifications
CAS Number
863491-70-7
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery, Protein Biochemistry
Smiles
C (NC1=NC2=C (C=C1) C=C (C (N[C@H] (C (N (CC3=CC=C (F) C=C3) C) =O) C4=CC=CC=C4) =O) C=C2) (=O) C5=C (C=CC=C5) C6=CC=C (OC (C) C) C=C6
Molecular Formula
C42H37FN4O4
Molecular Weight
680.77
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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