GLP-1R Antagonist 1
GLP-1R Antagonist 1 is a brain-penetrant, orally bioavailable small molecule that non-competitively inhibits the glucagon-like peptide 1 receptor with an IC50 of 650 nM. It is a valuable research tool for investigating GLP-1R signaling in metabolic and neurological studies, suitable for both in vitro assays and in vivo models.
Product Specifications
CAS Number
488097-06-9
Product Name Alternative
GLP-1R, GLP1R Antagonist 1, GLP-1R Antagonist 1, GLP 1R Antagonist 1, GLP-1, GlucagonReceptor, Glucagon Receptor
Field of Research
Pharmacology & Drug Discovery
Purity
90.00% (May vary between batches)
Solubility
10% DMSO+90% Corn Oil:3.3 mg/mL (7.49 mM) ; DMSO:90 mg/mL (204.21 mM)
Smiles
Cn1c2NC (=NC (c2c (=O) n (C) c1=O) (C (F) (F) F) C (F) (F) F) c1ccc (Cl) cc1
Molecular Formula
C16H11ClF6N4O2
Molecular Weight
440.73
Storage Conditions
-20°C
Notes
For research use only.
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