Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

GNE-207

GNE-207 is a potent, selective, and orally bioavailable CBP bromodomain inhibitor with an IC50 of 1 nM, demonstrating >2500-fold selectivity over BRD4. It effectively reduces MYC expression in MV-4-11 cells (EC50 = 18 nM) and is a valuable chemical probe for studying CBP/EP300 biology in cancer and other disease research.

Product Specifications

CAS Number

2158266-58-9

Field of Research

Epigenetics & Chromatin

Smiles

CNC (=O) c1ccc (cn1) -c1cc2cccc (-c3nn (C4CCOCC4) c4CCN (Cc34) C (C) =O) c2cn1

Molecular Formula

C29H30N6O3

Molecular Weight

510.59

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

STAT5 Rabbit Polyclonal Antibody (BF680)
orb1586296 100 µL

STAT5 Rabbit Polyclonal Antibody (BF680)

Sign In for Pricing
View Details
TMEM86A Protein Vector (Human) (pPM-C-His)
PV043040 500 ng

TMEM86A Protein Vector (Human) (pPM-C-His)

Sign In for Pricing
View Details
Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit
abx153980-01 96 Tests

Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit

Sign In for Pricing
View Details
Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit
abx153980-02 5x 96 Tests

Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit

Sign In for Pricing
View Details
Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit
abx153980-03 10x 96 Tests

Mouse Family With Sequence Similarity 135, Member B (FAM135B) ELISA Kit

Sign In for Pricing
View Details
Recombinant Chicken Cysteine and histidine-rich domain-containing protein 1 (CHORDC1)
MBS1469265-01 0.02 mg (E-Coli)

Recombinant Chicken Cysteine and histidine-rich domain-containing protein 1 (CHORDC1)

Sign In for Pricing
View Details