UPGL00004
UPGL00004 is a potent and selective glutaminase C (GAC) inhibitor, demonstrating high affinity with a Kd of 27 nM and inhibiting GAC activity with an IC50 of 29 nM. It effectively suppresses the proliferation of aggressive triple-negative breast cancer cells in vitro, making it a valuable tool for studying cancer metabolism and therapeutic targeting.
Product Specifications
CAS Number
1890169-95-5
Product Name Alternative
Glutaminase C, UPGL 00004, UPGL00004, UPGL-00004
Field of Research
Protein Biochemistry
Purity
97.44% (May vary between batches)
Solubility
DMSO:112.5 mg/mL (210.41 mM)
Smiles
O=C (Cc1ccccc1) Nc1nnc (NC2CCN (CC2) c2nnc (NC (=O) Cc3ccccc3) s2) s1
Molecular Formula
C25H26N8O2S2
Molecular Weight
534.66
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
K4684303 1.0 µg DNA
2310045N01Rik sgRNA CRISPR Lentivector (Mouse) (Target 2)
Sign In for Pricing
View Details