UPGL00004

UPGL00004 is a potent and selective glutaminase C (GAC) inhibitor, demonstrating high affinity with a Kd of 27 nM and inhibiting GAC activity with an IC50 of 29 nM. It effectively suppresses the proliferation of aggressive triple-negative breast cancer cells in vitro, making it a valuable tool for studying cancer metabolism and therapeutic targeting.

Product Specifications

CAS Number

1890169-95-5

Product Name Alternative

Glutaminase C, UPGL 00004, UPGL00004, UPGL-00004

Field of Research

Protein Biochemistry

Purity

97.44% (May vary between batches)

Solubility

DMSO:112.5 mg/mL (210.41 mM)

Smiles

O=C (Cc1ccccc1) Nc1nnc (NC2CCN (CC2) c2nnc (NC (=O) Cc3ccccc3) s2) s1

Molecular Formula

C25H26N8O2S2

Molecular Weight

534.66

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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