PF-4981517
PF-4981517 (CYP3cide) is a potent, time-dependent, and selective CYP3A4 inhibitor, with IC50 values of 0.03 μM, 17 μM, and 71 μM for CYP3A4, CYP3A5, and CYP3A7, respectively. It is a valuable chemical tool for in vitro studies to delineate the specific roles of CYP3A4 versus CYP3A5 in drug metabolism pathways.
Product Specifications
CAS Number
1390637-82-7
Product Name Alternative
CYP3cide, CYP3A4, PF 4981517, PF4981517, PF-4981517
Field of Research
Metabolism Research
Purity
99.77% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween-80+45% Saline:4 mg/mL (8.76 mM) ; DMSO:40 mg/mL (87.61 mM)
Smiles
Cc1ccc (cc1) -c1c (cnn1C) -c1nn (C) c2ncnc (N3CC[C@@H] (C3) N3CCCCC3) c12
Molecular Formula
C26H32N8
Molecular Weight
456.59
Storage Conditions
-20°C
Notes
For research use only.
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