G36
G36 is a potent and selective cell-permeable GPER antagonist, effectively blocking estrogen- and G-1-induced signaling (IC50 ~112-165 nM) without activity on ERα/ERβ. It is a valuable pharmacological tool used in vitro and in vivo to dissect GPER-specific functions in cancer, cardiovascular, and metabolic research.
Product Specifications
CAS Number
1392487-51-2
Product Name Alternative
G36, G-36, EstrogenReceptor, Estrogen Receptor, GPER, ERR, G 36
Field of Research
Metabolism Research
Purity
99.49% (May vary between batches)
Solubility
DMSO:55 mg/mL (133.39 mM)
Smiles
[H][C@]12CC=C[C@@]1 ([H]) c1cc (ccc1N[C@H]2c1cc2OCOc2cc1Br) C (C) C
Molecular Formula
C22H22BrNO2
Molecular Weight
412.32
Storage Conditions
-20°C
Notes
For research use only.
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