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PERK-IN-3

PERK-IN-3 is a highly potent and selective PERK inhibitor with an IC50 of 7.4 nM. This small molecule is a valuable research tool for investigating the unfolded protein response (UPR) in cellular and animal models of diseases such as cancer and neurodegeneration.

Product Specifications

CAS Number

1337532-08-7

Field of Research

Cell Biology, Signal Transduction

Smiles

NC1=C2C (=COC2=NC=N1) C=3C=C4C (=CC3) N (C (CC5=C (F) C=CC (F) =C5) =O) CC4

Molecular Formula

C22H16F2N4O2

Molecular Weight

406.38

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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