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GX-674

GX-674 is a potent and selective Nav1.7 channel blocker (IC50 = 0.1 nM at -40 mV) . It is a valuable research tool for investigating pain mechanisms, supporting both in vitro electrophysiology studies and in vivo models of inflammatory and neuropathic pain.

Product Specifications

CAS Number

1432913-36-4

Product Name Alternative

SodiumChannel, Sodium Channel, Nav1.7 channel, GX 674, GX674, GX-674

Field of Research

Pharmacology & Drug Discovery

Purity

98.60% (May vary between batches)

Solubility

DMSO:Soluble

Smiles

O (C1=C (C=C (Cl) C=C1) C=2C=C3C (=CC2) N=C (N) N3) C4=C (F) C=C (S (NC5=NC=NS5) (=O) =O) C (F) =C4

Molecular Formula

C21H13ClF2N6O3S2

Molecular Weight

534.95

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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