VUF-10497
VUF-10497 is a potent and selective inverse agonist of the histamine H4 receptor (pKi = 7.57) with demonstrated anti-inflammatory activity in rat models. It also exhibits significant affinity for the human histamine H1 receptor. This compound is a valuable pharmacological tool for studying histamine receptor signaling and inflammation in both in vitro and in vivo research.
Product Specifications
CAS Number
1080623-12-6
Field of Research
Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery
Smiles
N (CC1=CC=CS1) C=2C3=C (N=C (N2) N4CCN (C) CC4) C=CC (Cl) =C3
Molecular Formula
C18H20ClN5S
Molecular Weight
373.9
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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