Lomitapide Mesylate

Lomitapide Mesylate (BMS-201038 mesylate) is the mesylate salt form of lomitapide, a potent and selective small-molecule inhibitor of microsomal triglyceride transfer protein (MTP) . It is widely used in biochemical research to investigate lipid metabolism, including in vitro enzyme assays and in vivo models of dyslipidemia and homozygous familial hypercholesterolemia.

Product Specifications

CAS Number

202914-84-9

Product Name Alternative

MTP, Lomitapide, Lomitapide Mesylate, Inhibitor, inhibit, BMS 201038, BMS 201038 Mesylate, BMS201038, BMS-201038, BMS201038 Mesylate, BMS-201038 mesylate, BMS-201038 Mesylate, AEGR733, AEGR-733, AEGR733 Mesylate, AEGR-733 mesylate, AEGR-733 Mesylate, AEGR 733, AEGR 733 Mesylate

Field of Research

Metabolism Research, Pharmacology & Drug Discovery, Protein Biochemistry

Purity

99.65% (May vary between batches)

Solubility

10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (5.06 mM) ; DMSO:122 mg/mL (154.46 mM) ; Ethanol:93 mg/mL (117.75 mM) ; H2O:< 1 mg/mL (insoluble or slightly soluble)