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BKM-570

BKM-570 is a potent bradykinin B1 receptor antagonist that demonstrates significant antitumor activity. It has been shown to inhibit the growth of lung and prostate cancer models in both in vitro cell-based assays and in vivo animal studies, supporting its use in oncology research.

Product Specifications

CAS Number

259885-54-6

Field of Research

Pharmacology & Drug Discovery

Smiles

[C@H] (CC1=CC=C (OCC2=C (Cl) C=CC=C2Cl) C=C1) (C (NC3CC (C) (C) NC (C) (C) C3) =O) NC (C=CC4=C (F) C (F) =C (F) C (F) =C4F) =O

Molecular Formula

C34H34Cl2F5N3O3

Molecular Weight

698.55

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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