Elismetrep
Elismetrep (MT-8554) is a potent and orally bioavailable TRPM8 channel antagonist. It is utilized in preclinical research to investigate mechanisms of pain and thermoregulation, with studies exploring its potential for alleviating conditions like menopausal hot flashes in vivo.
Product Specifications
CAS Number
1400699-64-0
Product Name Alternative
MT 8554, MT8554, MT-8554, Elismetrep, TRPVChannel, TRPV Channel, TRP Channel, TRPM8, TRPChannel
Field of Research
Pharmacology & Drug Discovery
Purity
99.37% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (6.08 mM) ; DMSO:80 mg/mL (147.46 mM)
Smiles
O=C (O) C1=CC=C (C=C1) S (=O) (=O) N (C=2N=CC3=CC=CC=C3C2C4CC4) CC5=CC=C (OC (F) (F) F) C=C5
Molecular Formula
C27H21F3N2O5S
Molecular Weight
542.53
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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