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LP-471756

LP-471756 is a potent and selective GPR139 antagonist, effectively inhibiting LP-360924-stimulated cAMP production with an IC50 of 640 nM. This compound is a valuable research tool for investigating GPR139 receptor function in both in vitro and in vivo studies related to neuropharmacology and metabolic research.

Product Specifications

CAS Number

413605-11-5

Product Name Alternative

GPR139, LP 471756, LP471756, LP-471756

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Purity

99.59% (May vary between batches)

Solubility

DMSO:225 mg/mL (682.94 mM)

Smiles

Cc1ccccc1NS (=O) (=O) c1ccc (cc1) C1CCCCC1

Molecular Formula

C19H23NO2S

Molecular Weight

329.46

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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