LSN2814617
LSN2814617 is a potent, selective, and brain-penetrant mGlu5 positive allosteric modulator (PAM) with EC50 values of 52 nM (human) and 42 nM (rat) . In vivo studies indicate it promotes wakefulness with minimal rebound hypersomnolence, supporting its research application in neuropsychiatric conditions such as schizophrenia.
Product Specifications
CAS Number
1313498-17-7
Field of Research
Neuroscience
Smiles
C (C) (C) (C) C=1N2C (C[C@H] (CC2) C3=NC (=NO3) C4=CC=C (F) C=C4) =NN1
Molecular Formula
C18H20FN5O
Molecular Weight
341.38
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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