PD-217014 HCl
PD-217014 is a GABA analog that acts as a potent, nanomolar-affinity ligand (Ki = 18 nM) for the alpha-2-delta subunit of voltage-gated calcium channels, inhibiting gabapentin binding. It demonstrates visceral analgesic properties in vivo, making it a useful research tool for studying neuropathic pain and calcium channel function.
Product Specifications
CAS Number
444088-20-4
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
C (C (OC) =O) [C@@]1 (CN) C[C@@]2 ([C@] (C1) (CC2) [H]) [H]
Molecular Formula
C11H19NO2
Molecular Weight
197.27
Storage Conditions
-20°C
Notes
For research use only.
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