PF-04628935
PF-04628935 is a potent, orally bioavailable, and brain-penetrant ghrelin receptor (GHS-R1a) antagonist/inverse agonist with an IC50 of 4.6 nM. It is a valuable research tool for investigating the role of ghrelin signaling in metabolic disorders, appetite regulation, and related behaviors in both in vitro and in vivo models.
Product Specifications
CAS Number
1383719-97-8
Field of Research
Pharmacology & Drug Discovery
Smiles
C (N1CC2 (C1) CCN (C (CC3=CN4C (=N3) SC (C) =C4) =O) CC2) C5=C (Cl) C=C (C=C5) N6N=CC=N6
Molecular Formula
C24H26ClN7OS
Molecular Weight
496.03
Storage Conditions
-20°C
Notes
For research use only.
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