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PF-04628935

PF-04628935 is a potent, orally bioavailable, and brain-penetrant ghrelin receptor (GHS-R1a) antagonist/inverse agonist with an IC50 of 4.6 nM. It is a valuable research tool for investigating the role of ghrelin signaling in metabolic disorders, appetite regulation, and related behaviors in both in vitro and in vivo models.

Product Specifications

CAS Number

1383719-97-8

Field of Research

Pharmacology & Drug Discovery

Smiles

C (N1CC2 (C1) CCN (C (CC3=CN4C (=N3) SC (C) =C4) =O) CC2) C5=C (Cl) C=C (C=C5) N6N=CC=N6

Molecular Formula

C24H26ClN7OS

Molecular Weight

496.03

Storage Conditions

-20°C

Notes

For research use only.

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