MK761
MK761 is a dual-action small molecule combining β-adrenergic receptor blockade with vasodilation. Its antagonist efficacy is comparable to timolol and indololol, as demonstrated in vitro using isolated cat papillary muscle and rat atria. This profile supports cardiovascular research, including studies on hypertension and heart failure mechanisms.
Product Specifications
CAS Number
65321-41-7
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
O (C[C@H] (CNC (C) (C) C) O) C1=C (C#N) C=CC=N1
Molecular Formula
C13H19N3O2
Molecular Weight
249.31
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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