TP-238
TP-238 is a potent and selective dual CECR2/BPTF bromodomain inhibitor with respective IC50 values of 30 nM and 350 nM, and it also inhibits BRD9 (pIC50 5.9) . This probe compound is a valuable chemical tool for epigenetic research, enabling the study of chromatin remodeling and gene regulation in both cellular and biochemical assays.
Product Specifications
CAS Number
2415263-04-4
Field of Research
Epigenetics & Chromatin
Smiles
N (CCCN1C=CC=N1) C2=CC (=NC (S (C) (=O) =O) =N2) C3=CC=C (OCCCN (C) C) C=C3
Molecular Formula
C22H30N6O3S
Molecular Weight
458.58
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog