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PI3Kα-IN-4

PI3Kα-IN-4 is a highly potent and selective oral PI3Kα inhibitor with an IC50 of 1.8 nM. It is a valuable research tool for studying PI3Kα signaling in oncology, demonstrating antitumor efficacy in both cellular assays and in vivo xenograft models.

Product Specifications

CAS Number

2322293-83-2

Field of Research

Signal Transduction

Smiles

CNC (=O) [C@H] (C) Cn1cnc2ccc (cc2c1=O) -c1cnc (OC) c (NS (=O) (=O) c2ccc (F) cc2Cl) c1

Molecular Formula

C25H23ClFN5O5S

Molecular Weight

560

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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