KuWal151
This compound is a potent and selective CLK inhibitor, showing highest activity against CLK4 (IC50 = 28 nM) and minimal off-target effects. It demonstrates potent anti-proliferative activity in various cancer cell lines at subnanomolar concentrations in vitro, supporting its use in oncology research and kinase signaling studies.
Product Specifications
CAS Number
2341841-06-1
Smiles
O=C1NCC=2C=CC=3C (=CNC3C12) C=4C=CC=C (Cl) C4
Molecular Formula
C16H11ClN2O
Molecular Weight
282.72
Storage Conditions
-20°C
Notes
For research use only.
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