GSK2879552
GSK2879552 is an orally active, irreversible, and selective mechanism-based inhibitor of lysine-specific demethylase 1 (LSD1) . It exhibits antineoplastic activity and has been investigated in preclinical studies, including in vitro assays and in vivo models, for cancers such as small cell lung carcinoma and acute myeloid leukemia.
Product Specifications
CAS Number
1401966-69-5
Product Name Alternative
LSD1, GSK 2879552, GSK 2879552 HCl, GSK2879552, GSK-2879552, GSK2879552 2HCl, GSK2879552 2HCl, HistoneDemethylase, Histone Demethylase
Field of Research
Epigenetics & Chromatin
Purity
99.22% (May vary between batches)
Solubility
DMSO:27 mg/mL (74.08 mM) ; Ethanol:<1 mg/mL;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.49 mM)
Smiles
OC (=O) c1ccc (CN2CCC (CN[C@@H]3C[C@H]3c3ccccc3) CC2) cc1
Molecular Formula
C23H28N2O2
Molecular Weight
364.48
Storage Conditions
-20°C
Notes
For research use only.
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