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AS-99 TFA

AS-99 TFA is a potent and selective ASH1L histone methyltransferase inhibitor with anti-leukemic activity. It demonstrates efficacy in cellular assays by blocking proliferation and inducing apoptosis, and reduces leukemia burden in vivo through downregulation of MLL fusion target genes.

Product Specifications

CAS Number

3115178-55-4

Field of Research

Epigenetics & Chromatin, Immunology & Inflammation

Smiles

O=C (O) C (F) (F) F.O=C (NCC=1C=CC=2C (=CN (C2C1) C3CCN (CC3) S (=O) (=O) C (F) (F) F) C=4C=CC=C (C4) C (=S) N) C5CN (C) C5

Molecular Formula

C29H31F6N5O5S2

Molecular Weight

707.71

Storage Conditions

-20°C

Notes

For research use only.

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