CB2R PAM
CB2R PAM is an orally bioavailable positive allosteric modulator of the cannabinoid CB2 receptor. It potentiates agonist-stimulated G-protein activity in vitro and demonstrates efficacy in a murine neuropathic pain model, supporting research in analgesia and neuroinflammation.
Product Specifications
CAS Number
2244579-87-9
Product Name Alternative
CB2R, CB2R PAM, CannabinoidReceptor, Cannabinoid Receptor, Ec2la
Field of Research
Pharmacology & Drug Discovery
Purity
98.17% (May vary between batches)
Solubility
10% DMSO+90% Corn Oil:2 mg/mL (4.59 mM) ; DMSO:45 mg/mL (103.37 mM)
Smiles
N (C (=O) C1CCCCCC1) C=2C (=O) N (CC3=CC=C (F) C=C3) C=C (Br) C2C
Molecular Formula
C21H24BrFN2O2
Molecular Weight
435.33
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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