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RX-37

RX-37 is a highly selective and potent BET inhibitor, exhibiting low nanomolar affinity for BRD2/3/4. It demonstrates potent anti-proliferative activity in MLL-rearranged acute leukemia cell lines in vitro and has shown efficacy in relevant in vivo xenograft models, supporting its use in oncology research.

Product Specifications

CAS Number

1627715-60-9

Field of Research

Epigenetics & Chromatin

Smiles

CC1=C (C2=C3C=4C (NC3=CC=N2) =CC (=C (OC) C4) C=5C (C) =NOC5C) C (=NN1) C6CC6

Molecular Formula

C24H23N5O2

Molecular Weight

413.47

Storage Conditions

-20°C

Notes

For research use only.

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