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Chk1-IN-5

Chk1-IN-5 is a potent and selective Chk1 inhibitor that blocks its autophosphorylation. This compound has demonstrated efficacy in suppressing tumor growth in colon cancer xenograft models, supporting its use in oncology research for studying DNA damage response pathways both in vitro and in vivo.

Product Specifications

CAS Number

2120398-39-0

Field of Research

Cell Biology, Epigenetics & Chromatin

Smiles

O (CCCN) C1=C (C (OC) =CC (F) =C1) C2=CC (NC=3C=NC (C#N) =CN3) =NN2

Molecular Formula

C18H18FN7O2

Molecular Weight

383.38

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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