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8Br-HA

8Br-HA is a potent and selective inhibitor of the fragile histidine triad (FHIT) diadenosine triphosphatase, exhibiting an IC50 of 0.12 μM. It demonstrates anti-proliferative activity in vitro against HCC827 and H460 lung cancer cell lines, with GI50 values of 0.87 and 5.9 μM, respectively. This compound serves as a valuable chemical probe for investigating FHIT-related signaling pathways in cancer research.

Product Specifications

CAS Number

2937864-01-0

Storage Conditions

-20°C

Notes

For research use only.

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