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IGF-1R inhibitor-2

IGF-1R inhibitor-2 (example 121) is a selective small molecule inhibitor of the insulin-like growth factor-1 receptor. By blocking IGF-1R signaling, it can reverse oncogenic transformation and promote apoptosis in cancer cells, making it a valuable tool for studying IGF-1R biology in both in vitro and in vivo cancer research models.

Product Specifications

CAS Number

1116236-15-7

Field of Research

Immunology & Inflammation; Pharmacology & Drug Discovery, Signal Transduction

Smiles

COc1cc2CCN (C) Cc2cc1Nc1nc (Nc2cccc (F) c2C (N) =O) c2cc[nH]c2n1

Molecular Formula

C24H24FN7O2

Molecular Weight

461.501

Storage Conditions

-20°C

Notes

For research use only.

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