MS67
MS67 is a potent and selective WDR5 degrader (Kd = 63 nM) with demonstrated anticancer activity in cellular and animal models. It shows high specificity, exhibiting no off-target activity against methyltransferases, kinases, GPCRs, ion channels, or transporters, making it a valuable chemical probe for oncology and epigenetics research.
Product Specifications
CAS Number
2407452-77-9
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Smiles
C[C@H] (NC (=O) [C@@H]1C[C@@H] (O) CN1C (=O) [C@@H] (NC (=O) CNC (=O) c1ccc (F) c (c1) -c1ccc (N2C[C@H] (C) N (C) [C@H] (C) C2) c (NC (=O) c2c[nH]c (=O) cc2C (F) (F) F) c1) C (C) (C) C) c1ccc (cc1) -c1scnc1C
Molecular Formula
C52H59F4N9O7S
Molecular Weight
1030.14
Storage Conditions
-20°C
Notes
For research use only.
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