Clocinnamox mesylate
Clocinnamox mesylate is an irreversible, systemically active μ-opioid receptor antagonist with high affinity (apparent Ki values: μ=0.7 nM, δ=1.9 nM, κ=5.7 nM in mice) . It is a valuable research tool for investigating opioid receptor function and mechanisms of antagonism in both in vitro binding assays and in vivo pharmacological studies.
Product Specifications
CAS Number
117332-69-1
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Smiles
CS (O) (=O) =O.[H][C@@]12Oc3c4c (C[C@@]5 ([H]) N (CC6CC6) CC[C@@]14[C@]5 (CCC2=O) NC (=O) C=Cc1ccc (Cl) cc1) ccc3O |w:30.33, TLB:8:9:22:14.19.20, THB:39:10:22:14.19.20|
Molecular Formula
C30H33ClN2O7S
Molecular Weight
601.11
Storage Conditions
-20°C
Notes
For research use only.
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