GP 1a
GP 1a is a potent and selective CB2 receptor agonist (EC50=7.1 nM) with demonstrated efficacy in cellular assays, including cAMP inhibition and ERK1/2 phosphorylation. It exhibits anti-inflammatory and anti-fibrotic properties, promoting epithelial regeneration, which supports its research application in models of skin wound healing and tissue repair.
Product Specifications
CAS Number
511532-96-0
Product Name Alternative
GP 1a, CB2, Cannabinoid Receptor, CannabinoidReceptor, PERK
Field of Research
Cell Biology, Pharmacology & Drug Discovery, Signal Transduction
Purity
99.44% (May vary between batches)
Solubility
Ethanol:90 mg/mL (203.92 mM) ; DMSO:90 mg/mL (203.92 mM)
Smiles
C (NN1CCCCC1) (=O) C=2C3=C (N (N2) C4=C (Cl) C=C (Cl) C=C4) C=5C (C3) =CC (C) =CC5
Molecular Formula
C23H22Cl2N4O
Molecular Weight
441.35
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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