Edg-2 receptor inhibitor 1
SAR-100842 is a potent and selective inhibitor of the Edg-2 (LPA1) receptor with an IC50 of <0.1 μM. This small molecule is a valuable research tool for investigating lysophosphatidic acid (LPA) signaling in fibrosis, neuropathic pain, and cancer research using both in vitro and in vivo models.
Product Specifications
CAS Number
1195941-38-8
Product Name Alternative
Edg 2 receptor inhibitor 1, EDG2, Edg2 receptor inhibitor 1, Edg-2 receptor inhibitor 1, LPA Receptor, LPAReceptor, SAR 100842, SAR100842, SAR-100842
Field of Research
Pharmacology & Drug Discovery
Purity
99.47% (May vary between batches)
Solubility
DMSO:83.3 mg/mL (186.98 mM)
Smiles
N (C (=O) C1=CC (OCCC2=CC (C) =CC=C2) =C (OC) C=C1) C3 (C (O) =O) CC=4C (C3) =CC=CC4
Molecular Formula
C27H27NO5
Molecular Weight
445.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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