Cis-4-Br-2,5-F2-PCPA
Cis-4-Br-2,5-F2-PCPA (S1024) is a potent inhibitor of LSD1 (Ki=94 nM) with selectivity over LSD2 (Ki=8.4 μM) . It suppresses cancer cell proliferation, as demonstrated in CCRF-CEM cells, by increasing global H3K4me2 levels. This compound is a useful research tool for studying epigenetic regulation in oncology and cancer stem cell biology.
Product Specifications
Field of Research
Epigenetics & Chromatin
Molecular Formula
C9H8BrF2N
Molecular Weight
248.07
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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