GAT564
GAT564 (Compound 15d) is a potent allosteric CB1 receptor modulator, enhancing orthosteric ligand binding with EC50 values of 87 nM (cAMP) and 320 nM (β-arrestin2) . It has demonstrated significant topical efficacy in reducing intraocular pressure in a murine glaucoma model, supporting research in cannabinoid receptor pharmacology and ocular therapeutics.
Product Specifications
Field of Research
Pharmacology & Drug Discovery
Molecular Formula
C20H16N2O2S
Molecular Weight
348.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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