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BRD4 Inhibitor-17

BRD4 Inhibitor-17 (Compound 5i) is a potent BRD4 inhibitor (IC50 = 0.33 μM) that regulates transcription of inflammatory and proliferative genes. Research indicates its utility in oncology and inflammation studies, with in vitro and in vivo models suggesting potential as an antidote for arsenical toxicity.

Product Specifications

Field of Research

Epigenetics & Chromatin, Epigenetics & Chromatin; Pharmacology & Drug Discovery

Molecular Formula

C16H16FN3O3S

Molecular Weight

349.38

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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