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AKN-028 acetate

AKN-028 acetate is a potent and orally bioavailable FLT3 tyrosine kinase inhibitor (IC50 = 6 nM) that blocks autophosphorylation. It demonstrates dose-dependent cytotoxicity and induces caspase-3-mediated apoptosis in vitro, supporting its research application in models of acute myeloid leukemia (AML) .

Product Specifications

Field of Research

Cardiovascular Research, Cell Biology, Protein Biochemistry, Signal Transduction

Molecular Formula

C19H18N6O2

Molecular Weight

362.39

Storage Conditions

-20°C

Notes

For research use only.

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