Bromodomain inhibitor-10
Bromodomain inhibitor-10 (compound 128) is a potent, dual-bromodomain inhibitor with high affinity for BRD4-1 (Kd=15 nM) and BRD4-2 (Kd=2500 nM) . It suppresses IL12p40 production and is a valuable chemical probe for epigenetic and inflammation research in cellular and biochemical assays.
Product Specifications
CAS Number
1870849-58-3
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Smiles
C (NC=1C=C2C (=CC1) NC (=O) C=C2C) (=O) C3=C (N=CC=C3) N4CCOCC4
Molecular Formula
C20H20N4O3
Molecular Weight
364.4
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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