MPT0G211 mesylate
MPT0G211 mesylate is a highly potent and orally bioavailable HDAC6 inhibitor with exceptional isoform selectivity (>1000-fold) and blood-brain barrier penetration. It has demonstrated efficacy in preclinical Alzheimer's disease models by reducing tau pathology and cognitive deficits, and also shows potential in cancer research for its anti-metastatic effects.
Product Specifications
CAS Number
2151854-33-8
Field of Research
Epigenetics & Chromatin, Molecular Biology
Smiles
CS (O) (=O) =O.ONC (=O) c1ccc (CNc2cccc3cccnc23) cc1
Molecular Formula
C18H19N3O5S
Molecular Weight
389.43
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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