AMG8788
AMG8788 is a potent, selective, and orally bioavailable antagonist of the TRPM8 ion channel, exhibiting an IC50 of 63.2 nM. This compound is a valuable research tool for investigating TRPM8's role in vivo and in vitro, particularly in areas such as cold sensation, migraine, and urological disorders.
Product Specifications
CAS Number
1159996-43-6
Field of Research
Pharmacology & Drug Discovery
Smiles
C (NC1=CC=C (F) C=C1) (=O) N2[C@@H] (C=3C (CC2) =CC=CC3) C4=CC=C (C (F) (F) F) C=C4
Molecular Formula
C23H18F4N2O
Molecular Weight
414.4
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
JOT-AP00099-01 20 µL
IGF-I Receptor beta(Phospho-Tyr1131) Rabbit Polyclonal Antibody
Sign In for Pricing
View Details JOT-AP00099-02 50 μL
IGF-I Receptor beta(Phospho-Tyr1131) Rabbit Polyclonal Antibody
Sign In for Pricing
View Details JOT-AP00099-03 100 µL
IGF-I Receptor beta(Phospho-Tyr1131) Rabbit Polyclonal Antibody
Sign In for Pricing
View Details 
E45O55039M2-100 100 µg
SARS-CoV-2 (2019-nCoV) Spike RBD (Y508H) -His Recombinant Protein
Sign In for Pricing
View Details TL304801V 500 µL Each
ELAC1 Human shRNA Lentiviral Particle (Locus ID 55520)
Sign In for Pricing
View Details