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CDK-IN-9

CDK-IN-9 (compound 24) is a potent, low-nanomolar CDK2/E inhibitor that also functions as a molecular gel to induce a CDK12-DDB1 interaction. This compound promotes the dephosphorylation of retinoblastoma protein and RNA polymerase II, leading to apoptosis, and is used in cancer research for studying cell cycle regulation and transcription.

Product Specifications

Field of Research

Cell Biology, Molecular Biology

Molecular Formula

C21H24N8S

Molecular Weight

420.53

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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