KDM1/CDK1-IN-1
KDM1/CDK1-IN-1 is a dual inhibitor of KDM1 and CDK1 with sub-micromolar potency. It induces G2/M cell cycle arrest and apoptosis, demonstrating cytotoxic effects in various cancer cell lines such as CCRF-CEM, HOP-92, and Hep-G2. This compound is a useful chemical probe for oncology research, particularly in studying cell cycle regulation and epigenetic modulation in vitro.
Product Specifications
Field of Research
Cell Biology, Epigenetics & Chromatin, Metabolism Research; Cell Biology, Protein Biochemistry
Molecular Formula
C22H17N5O3S
Molecular Weight
431.47
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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